iphepha_ibhena

Ishishini lePharmasuatical

Ishishini lePharmasuatical

I-amino acid ineempawu zokusabela ezininzi, ezinokuthi zisetyenziswe njengosetyenziso olubanzi lwemithombo yesandla kunye nokuhlanganiswa kweekhompawundi ezisekelwe ngesandla.Sisandla sendalo esikhoyo esona sigaba sibalulekileyo ngokwesondo.Ii-amino acids kwi-synthesis yamachiza zihlala zicatshulwa kwiimolekyuli zamachiza kwimodyuli yesakhiwo semolekyuli yamachiza, ukuqala ngesondo, okanye ukuhlanganiswa kwamachiza ezandla njenge-arhente yokukhubazeka.

Anti-hypertension
I-Hypertension iye yaba sesona siganeko sesifo senhliziyo kwisifo senhliziyo yabantu, kwaye sesona sizathu sibalulekileyo somngcipheko wezifo zentliziyo kunye ne-cerebrovascular.

Amayeza okubulala iintsholongwane
Amayeza okubulala iintsholongwane eCarbon moldyne ngamayeza okubulala iintsholongwane e-β-lactam aneyona spectrum yokulwa ne-antibacterial kunye nowona msebenzi unamandla wokulwa neebhaktiriya, kuba ine-tiimpawu zozinzo lwe-β-lactamase kunye netyhefu ephantsi ziye zaba zezona zibalulekileyo zamachiza okulwa ne-antibacterial ukunyanga usulelo olubi lwebhaktiriya-.

Anti-HIV
I-HIV protease inhibitors yenye yeendidi ezintathu zamachiza alwa ne-HIV, anokuthintela ngokufanelekileyo ukuphindaphinda kwentsholongwane kwaye ibe nguGawulayo.ain amayeza.

Ishishini lePharmasuatical

I-Antitumor
I-Classic dihydrocarbonic acid yokunciphisa i-enzyme inhibitors (i-aminotate, i-aminotrexate, i-Edutantis, i-Permeusceri) kunye ne-thymotide.I-synthetic enzymes inqanda iLeartisa equkethe i-L-glutamic acid intsalela isakhiwo.Indima ephambili kukwenza i-polymerization ye-polymerization ye-glutamate synthetase emzimbeni.
Ngohlobo lwepolymerization, uhlobo lwepolymerization ye-glutamic acid yonyusa ixesha lokugcinwa kweemolekyuli zamachiza kwiseli, ngaloo ndlela iphucula amandla ayo.inhibitory effect ye-hydrogen folic acid yokunciphisa i-enzyme.I-L-glutamic acid yinto ebalulekileyo ekrwada kwi-synthetic amayeza anjalo.